Thaum feem ntau siv rau tib lub ntsiab lus, GABA thiab Gabapentin yog cov chaw sib txawv nrog qhov sib txawv tseem ceeb thiab zoo sib xws. Cov lus qhia dav dav no nkag mus tob rau hauv lawv cov yam ntxwv thiab tshawb nrhiav lawv txoj kev sib raug zoo kom paub meej txog qhov tsis meej pem.
GABA: Lub Ntuj Inhibitory Neurotransmitter
GABA, luv luv rau gamma-aminobutyric acid, yog thawj inhibitory neurotransmitter hauv nruab nrab paj hlwb (CNS). Nws ua lub luag haujlwm tseem ceeb hauv kev tswj hwm kev ua haujlwm neuronal, txo qis excitation, thiab txhawb kev so. Los ntawm kev khi rau cov receptors tshwj xeeb hauv lub hlwb, GABA inhibits neurons firing, ua rau kom muaj kev ntxhov siab thiab txhawb kev pw tsaug zog.
Kev ua haujlwm ntawm GABA
Txo kev ntxhov siab thiab kev ntxhov siab:GABA cov nyhuv calming pab tswj kev ntxhov siab thiab kev ntxhov siab los ntawm inhibiting overactive neurons nyob rau hauv lub hlwb.
Txhim kho pw tsaug zog:GABA pab txhawb kev pw tsaug zog pib thiab tswj kev pw tsaug zog zoo los ntawm kev txhawb nqa kev so thiab txo lub hlwb ua haujlwm.
Txo qhov mob pom:GABA plays lub luag haujlwm hauv kev tswj qhov mob los ntawm kev hloov pauv kev sib kis ntawm cov cim mob hauv qaum qaum.
Txhawb kev txawj ntse muaj nuj nqi:GABA tuaj yeem pab txhawb kev txawj ntse los ntawm kev txhim kho kev nco, kev kawm, thiab kev xav.
GABA Deficiency thiab lwm yam mob
Qib qis ntawm GABA tau cuam tshuam nrog ntau yam mob, suav nrog:
Kev ntxhov siab vim
Kev nyuaj siab
Insomnia
Epilepsy
Mob mob
ADHD
Gabapentin: Ib qho Mimic ntawm GABA's Effects
Gabapentin yog ib hom tshuaj uas tau muab cais ua GABA analog. Thaum tsis zoo ib yam rau GABA, nws qhia qee qhov zoo sib xws thiab cuam tshuam nrog lub paj hlwb hauv txoj hauv kev uas ua rau cov teebmeem ntawm GABA. Txawm hais tias qhov tseeb mechanism ntawm kev txiav txim tseem tab tom tshawb nrhiav, Gabapentin tau ntseeg tias ua haujlwm los ntawm:
Kev khi rau alpha-2-delta subunits ntawm voltage-gated calcium channel tiv thaiv kev tso tawm ntawm excitatory neurotransmitters.
Inhibiting lub reuptake ntawm GABA, yog li nce nws concentration nyob rau hauv lub synaptic cleft.
Kev Siv Tshuaj Kho Mob ntawm Gabapentin
Epilepsy:Gabapentin tau pom zoo raws li kev kho mob ntxiv rau qee qhov qaug dab peg hauv cov neeg laus thiab menyuam yaus.
Neuropathic mob:Nws muaj txiaj ntsig zoo hauv kev tswj cov mob uas cuam tshuam nrog cov paj hlwb puas, xws li mob ntshav qab zib neuropathy, postherpetic neuralgia, thiab trigeminal neuralgia.
Restless Leg Syndrome (RLS):Gabapentin pab txo qis cov tsos mob ntawm RLS, suav nrog kev tsis tuaj yeem txav ceg thiab pw tsaug zog.
Kub flashes:Cov kev tshawb fawb tsis ntev los no qhia tias gabapentin tuaj yeem txo qhov kub nyhiab cuam tshuam nrog kev ua haujlwm tsis zoo.
Gabapentin vs. GABA: Qhov txawv tseem ceeb
Nov yog cov lus qhia txog qhov sib txawv tseem ceeb ntawm GABA thiab Gabapentin:
| Feature | GABA | Gabapentin |
|---|---|---|
| Xwm | Ntuj neurotransmitter | Synthetic tshuaj |
| Qauv | Amino acid | Cyclic amino acid derivative |
| Mechanism ntawm kev ua | Txuas rau GABA receptors | Mimics cov teebmeem ntawm GABA |
| Qhov chaw | Tsim nyob rau hauv lub hlwb | Tsim nyob rau hauv ib lub chaw kuaj |
| Muaj | Ntuj tshwm sim | Yuav tsum tau muab tshuaj |
| Siv | Ntau yam ntawm physiological functions | Kev kho mob tshwj xeeb |
| Kev mob tshwm sim | Feem ntau zoo zam | tuaj yeem ua rau qaug zog, kiv taub hau, thiab qaug zog |
Zoo sib xws ntawm GABA thiab Gabapentin
Ob leeg txhawb kev so thiab txo kev ntxhov siab.
Ob leeg muaj peev xwm siv tau los tswj qhov mob thiab pw tsaug zog tsis zoo.
Ob leeg cuam tshuam nrog lub paj hlwb los hloov kho cov haujlwm neuronal.
Kev txiav txim siab tseem ceeb
Thaum Gabapentin ua raws li cov teebmeem ntawm GABA, nws tsis yog qhov hloov pauv ncaj qha. Nws yog ib qho tseem ceeb kom sab laj nrog kws kho mob ua ntej noj Gabapentin, tshwj xeeb tshaj yog tias koj muaj mob hauv qab los yog noj lwm yam tshuaj. Tsis tas li ntawd, nco ntsoov tias Gabapentin tuaj yeem muaj kev phiv, yog li nws tseem ceeb heev kom paub txog lawv thiab tham nrog koj tus kws kho mob.
Kev taw qhia yav tom ntej
Kev tshawb fawb rau GABA thiab Gabapentin txuas ntxiv tshawb nrhiav lawv cov kev siv peev xwm hauv ntau qhov chaw kho mob. Kev nkag siab txog lawv cov kev cuam tshuam nrog lub paj hlwb thiab lawv qhov cuam tshuam rau cov xwm txheej sib txawv tuaj yeem ua rau muaj kev txhim kho ntau lub hom phiaj thiab kev kho mob zoo rau qaug dab peg, mob, thiab lwm yam kab mob neurological.
Xaus
GABA thiab Gabapentin, txawm hais tias cov chaw sib txawv muaj lub hom phiaj sib xws: txhawm rau txhawb kom muaj kev thaj yeeb nyab xeeb thiab tswj hwm kev ua haujlwm neuronal. Thaum GABA yog ib qho kev hloov pauv hauv lub cev nrog ntau lub zog, Gabapentin yog cov tshuaj hluavtaws uas ua rau qee yam ntawm nws cov teebmeem rau kev kho mob tshwj xeeb. Kev nkag siab txog lawv tus yam ntxwv thiab kev sib raug zoo uas lawv sib koom yog qhov tseem ceeb rau kev sib tham txog lawv lub luag haujlwm hauv kev noj qab haus huv thiab kev noj qab haus huv.
Cov ntaub ntawv no, ntau tshaj 1000 lo lus, lub hom phiaj los muab cov ntsiab lus dav dav ntawm GABA thiab Gabapentin thiab qhia meej txog cov kev xav tsis zoo. Thov nco ntsoov, qhov no tsis yog los hloov cov lus qhia kev kho mob. Nco ntsoov sab laj nrog koj tus kws kho mob kom paub qhov tseeb thiab cov kev kho mob tsim nyog.
Cov ntaub ntawv:
https://astrasama.com/difference-between-gaba-and-gabapentin/
